| 2026 | Yang, Haijian and Dong, Wenyan and An, Yana and He, Zhanyu and Pan, Hui and Pan, Wencong and Tan, Jianhui and Sun, Jingjing and Shen, Chuan and Su, Wu and others: Ansamer-Controlled Bicyclic Peptides as Integrin $\alpha$v$\beta$6 Targeting Agents. In: Angewandte Chemie International Edition, 65, 2026, e1254428 |
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| 2026 | Tian, Hui and Pan, Wencong and Shi, Huaihuai and Shao, Ximing and Sun, Jingjing and Liang, Jiaming and Chen, Bichun and Cheng, Binghua and Liu, Ke and Yao, Guiyang and others: Coibamide analogue as a novel-class payload for antibody-drug conjugate. In: Journal of Medicinal Chemistry, 69, 2026, 5691--5702 |
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| 2026 | Yang, Haijian and Pan, Hui and Ran, Ting and Dong, Wenyan and Pan, Wencong and Tan, Jianhui and Sun, Jingjing and Süssmuth, Roderich D and Su, Wu and Yao, Guiyang: Identification of an $\alpha$v$\beta$3-targeting bicyclic peptide with atypical nor Arg-Gly-Asp sequence. In: Communications Chemistry, 9, 2026, 83 |
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| 2026 | Hao, Qingqing and Wang, Laurie and Pan, Hui and Xiao, Xihui and Dong, Wenyan and Pan, Wencong and Sun, Jingjing and Su, Wu and Fang, Lijing and Park, Eunyong and others: Structure-based design of Sec61 translocon targeting prodrugs minimize off-target toxicity. In: Cell Chemical Biology, 33, 2026, 823--836 |
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| 2026 | He, Zhanyu and Janssen, Celine and Schäfer, Joana-Lysiane and Mühlenweg, Agnes and Kosol, Simone and Jarling, Rene and Mainz, Andi and Keller, Bettina G and Yao, Guiyang and Klussmann, Enno and others: Synthesis and characterization of cortinarins--cryptic cyclic peptides from mushrooms of the genus Cortinarius. In: Chemical Science, 2026, |
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| 2025 | Zhou, Yi and Jin, Jingyan and Zhou, Pingzheng and Su, Wu and Yao, Guiyang: Adding AC-Terminal Amino Acid Prevents the Conformational Interconversion of Plecantide Analogs. In: ChemBioChem, 26, 2025, e202500237 |
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| 2025 | Wang, Chaoming and Zhang, Jing and Wang, Dongping and Chen, Shengle and Yuan, Qi and Yin, Ruijuan and Yao, Guiyang and Qi, Xin and Li, Jing and Jiang, Tao: Conjugating 10, 11-Dimethoxy-camptothecin with an Integrin $\alpha$v$\beta$3-Targeting Peptide through a Triazine Linker for Targeted Tumor Treatment in Lung and Pancreatic Carcinoma. In: Journal of Medicinal Chemistry, 68, 2025, 25091--25111 |
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| 2025 | Chen, Bichun and Bai, Jinyu and Shi, Huaihuai and Hao, Rui and Liang, Jiaxin and Tian, Hui and Yao, Guiyang and Shao, Ximing and Li, Hongchang and Wang, Ruibing and others: Degrader-drug conjugate (DDC) mediated immunochemotherapy for tumor treatment. In: Journal of Medicinal Chemistry, 68, 2025, 26218--26233 |
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| 2024 | Gonzalez, Barbara Daiana and Forbrig, Enrico and Yao, Guiyang and Kielb, Patrycja and Mroginski, Maria Andrea and Hildebrandt, Peter and Kozuch, Jacek: Cation Dependence of Enniatin B/Membrane-Interactions Assessed Using Surface-Enhanced Infrared Absorption (SEIRA) Spectroscopy. In: ChemPlusChem, 89, 2024, e202400159 |
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| 2024 | Sehit, Ekin and Yao, Guiyang and Battocchio, Giovanni and Radfar, Rahil and Trimpert, Jakob and Mroginski, Maria A and Süssmuth, Roderich and Altintas, Zeynep: Computationally designed epitope-mediated imprinted polymers versus conventional epitope imprints for the detection of human adenovirus in water and human serum samples. In: ACS sensors, 9, 2024, 1831--1841 |
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| 2024 | Sehit, Ekin and Yao, Guiyang and Battocchio, Giovanni and Radfar, Rahil and Trimpert, Jakob and Mroginski, Maria A and Süssmuth, Roderich and Altintas, Zeynep: Computationally designed epitope-mediated imprinted polymers versus conventional epitope imprints for the detection of human adenovirus in water and human serum samples. In: ACS sensors, 9, 2024, 1831--1841 |
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| 2022 | Utesch, Tillmann and Staffa, Jana and Katz, Sagie and Yao, Guiyang and Kozuch, Jacek and Hildebrandt, Peter: Potential distribution across model membranes. In: The Journal of Physical Chemistry B, 126, 2022, 7664--7675 |
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| 2022 | Wenz, Marius T and Kosol, Simone and Yao, Guiyang and Süssmuth, Roderich D and Keller, Bettina G: The influence of N-methylation on the ansamers of an amatoxin: Gly5Sar-amanullin. In: bioRxiv, 2022, 2022--12 |
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| 2022 | Yao, Guiyang and Kosol, Simone and Wenz, Marius T and Irran, Elisabeth and Keller, Bettina G and Trapp, Oliver and Süssmuth, Roderich D: The occurrence of ansamers in the synthesis of cyclic peptides. In: Nature Communications, 13, 2022, 6488 |
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| 2022 | Yao, Guiyang and Kosol, Simone and Wenz, Marius T and Irran, Elisabeth and Keller, Bettina G and Trapp, Oliver and Süssmuth, Roderich D: The occurrence of ansamers in the synthesis of cyclic peptides. In: Nature Communications, 13, 2022, 6488 |
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| 2021 | Yao, Guiyang and Knittel, Caroline H and Kosol, Simone and Wenz, Marius T and Keller, Bettina G and Gru{\ss}, Hendrik and Braun, Alexandra C and Lutz, Christian and Hechler, Torsten and Pahl, Andreas and others: Iodine-mediated tryptathionine formation facilitates the synthesis of amanitins. In: Journal of the American Chemical Society, 143, 2021, 14322--14331 |
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| 2021 | Yao, Guiyang and Knittel, Caroline H and Kosol, Simone and Wenz, Marius T and Keller, Bettina G and Gru{\ss}, Hendrik and Braun, Alexandra C and Lutz, Christian and Hechler, Torsten and Pahl, Andreas and others: Iodine-mediated tryptathionine formation facilitates the synthesis of amanitins. In: Journal of the American Chemical Society, 143, 2021, 14322--14331 |
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| 2021 | Qin, Feng and Wang, Cai Yi and Kim, Donghwa and Wang, Heng-Shan and Zhu, Yan-Kui and Lee, Sang Kook and Yao, Gui-Yang and Liang, Dong: Nitidumpeptins A and B, cyclohexapeptides isolated from Zanthoxylum nitidum var. tomentosum: structural elucidation, total synthesis, and antiproliferative activity in cancer cells. In: The Journal of Organic Chemistry, 86, 2021, 1462--1470 |
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| 2021 | Qin, Feng and Wang, Cai Yi and Kim, Donghwa and Wang, Heng-Shan and Zhu, Yan-Kui and Lee, Sang Kook and Yao, Gui-Yang and Liang, Dong: Nitidumpeptins A and B, cyclohexapeptides isolated from Zanthoxylum nitidum var. tomentosum: structural elucidation, total synthesis, and antiproliferative activity in cancer cells. In: The Journal of Organic Chemistry, 86, 2021, 1462--1470 |
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| 2019 | Yao, Guiyang and Joswig, Jan-Oliver and Keller, Bettina G and Süssmuth, Roderich D: Total Synthesis of the Death Cap Toxin Phalloidin: Atropoisomer Selectivity Explained by Molecular-Dynamics Simulations. In: Chemistry--a European Journal, 25, 2019, 8030--8034 |
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| 2019 | Yao, Guiyang and Joswig, Jan-Oliver and Keller, Bettina G and Süssmuth, Roderich D: Total Synthesis of the Death Cap Toxin Phalloidin: Atropoisomer Selectivity Explained by Molecular-Dynamics Simulations. In: Chemistry--a European Journal, 25, 2019, 8030--8034 |
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| 2018 | Yao, Guiyang and Wang, Wei and Ao, Lijiao and Cheng, Zhehong and Wu, Chunlei and Pan, Zhengyin and Liu, Ke and Li, Hongchang and Su, Wu and Fang, Lijing: Improved total synthesis and biological evaluation of coibamide A analogues. In: Journal of medicinal chemistry, 61, 2018, 8908--8916 |
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| 2018 | Yao, Guiyang and Wang, Wei and Ao, Lijiao and Cheng, Zhehong and Wu, Chunlei and Pan, Zhengyin and Liu, Ke and Li, Hongchang and Su, Wu and Fang, Lijing: Improved total synthesis and biological evaluation of coibamide A analogues. In: Journal of medicinal chemistry, 61, 2018, 8908--8916 |
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| 2018 | Li, De-zhi and Han, Bing-nan and Wei, Rui and Yao, Gui-yang and Chen, Zhizhen and Liu, Jie and Poon, Terence CW and Su, Wu and Zhu, Zhongyu and Dimitrov, Dimiter S and others: N-terminal $\alpha$-amino group modification of antibodies using a site-selective click chemistry method. MAbs. 2018. 712--719 |
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| 2018 | Li, De-zhi and Han, Bing-nan and Wei, Rui and Yao, Gui-yang and Chen, Zhizhen and Liu, Jie and Poon, Terence CW and Su, Wu and Zhu, Zhongyu and Dimitrov, Dimiter S and others: N-terminal $\alpha$-amino group modification of antibodies using a site-selective click chemistry method. MAbs. 2018. 712--719 |
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| 2017 | Tan, Yuanyan and Wang, Wei and Wu, Chunlei and Pan, Zhengyin and Yao, Guiyang and Fang, Lijing and Su, Wu: Myristic acid-modified thymopentin for enhanced plasma stability and immune-modulating activity. In: International immunopharmacology, 47, 2017, 88--94 |
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| 2017 | Huang, Ri-zhen and Jin, Le and Yao, Gui-yang and Dai, Wei-long and Huang, Xiao-chao and Liao, Zhi-Xin and Wang, Heng-shan: Synthesis and molecular docking study of novel alizarin derivatives containing phosphoryl amino acid moiety as potential antitumor agents. In: Medicinal Chemistry Research, 26, 2017, 2363--2374 |
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| 2017 | Wu, Chunlei and Pan, Zhengyin and Yao, Guiyang and Wang, Wei and Fang, Lijing and Su, Wu: Synthesis and structure--activity relationship studies of teixobactin analogues. In: Rsc Advances, 7, 2017, 1923--1926 |
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| 2017 | Wu, Chunlei and Pan, Zhengyin and Yao, Guiyang and Wang, Wei and Fang, Lijing and Su, Wu: Synthesis and structure--activity relationship studies of teixobactin analogues. In: Rsc Advances, 7, 2017, 1923--1926 |
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| 2017 | Qin, Jian-Mei and Huang, Ri-Zhen and Yao, Gui-Yang and Liao, Zhi-Xin and Pan, Ying-Ming and Wang, Heng-Shan: Terminal functionalized thiourea-containing dipeptides as multidrug-resistance reversers that target 20S proteasome and cell proliferation. In: European Journal of Medicinal Chemistry, 126, 2017, 259--269 |
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| 2017 | Zhengyin, Pan and Chunlei, Wu and Wei, Wang and Zhehong, Cheng and Guiyang, Yao and Ke, Liu and Hongchang, Li and Lijing, Fang and Wu, Su: Total Synthesis and Stereochemical Assignment of Gymnopeptides A and B. 2017, |
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| 2017 | Pan, Zhengyin and Wu, Chunlei and Wang, Wei and Cheng, Zhehong and Yao, Guiyang and Liu, Ke and Li, Hongchang and Fang, Lijing and Su, Wu: Total synthesis and stereochemical assignment of gymnopeptides A and B. In: Organic letters, 19, 2017, 4420--4423 |
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| 2016 | Yao, Guiyang and Ye, Manyi and Zhu, Yongtao and Liao, Zhixin and Wang, Hengshan: Synthesis and pharmacological evaluation of maleopimaric N-arylimides: Identification of novel proapoptotic agents. In: Anti-Cancer Agents in Medicinal Chemistry-Anti-Cancer Agents), 16, 2016, 755--762 |
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| 2016 | Huang, Ri-Zhen and Wang, Cai-Yi and Li, Jian-Fei and Yao, Gui-Yang and Pan, Ying-Ming and Ye, Man-Yi and Wang, Heng-Shan and Zhang, Ye: Synthesis, antiproliferative and apoptosis-inducing effects of novel asiatic acid derivatives containing $\alpha$-aminophosphonates. In: RSC advances, 6, 2016, 62890--62906 |
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| 2016 | Huang, Ri-Zhen and Wang, Cai-Yi and Li, Jian-Fei and Yao, Gui-Yang and Pan, Ying-Ming and Ye, Man-Yi and Wang, Heng-Shan and Zhang, Ye: Synthesis, antiproliferative and apoptosis-inducing effects of novel asiatic acid derivatives containing $\alpha$-aminophosphonates. In: RSC advances, 6, 2016, 62890--62906 |
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| 2015 | Hua, Shi-Xian and Huang, Ri-Zhen and Ye, Man-Yi and Pan, Ying-Ming and Yao, Gui-Yang and Zhang, Ye and Wang, Heng-Shan: Design, synthesis and in vitro evaluation of novel ursolic acid derivatives as potential anticancer agents. In: European Journal of Medicinal Chemistry, 95, 2015, 435--452 |
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| 2015 | Hua, Shi-Xian and Huang, Ri-Zhen and Ye, Man-Yi and Pan, Ying-Ming and Yao, Gui-Yang and Zhang, Ye and Wang, Heng-Shan: Design, synthesis and in vitro evaluation of novel ursolic acid derivatives as potential anticancer agents. In: European Journal of Medicinal Chemistry, 95, 2015, 435--452 |
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| 2015 | Guiyang, Yao and Zhengyin, Pan and Chunlei, Wu and Wei, Wang and Lijing, Fang and Wu, Su: Efficient Synthesis and Stereochemical Revision of Coibamide A. 2015, |
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| 2015 | Yao, Guiyang and Pan, Zhengyin and Wu, Chunlei and Wang, Wei and Fang, Lijing and Su, Wu: Efficient synthesis and stereochemical revision of coibamide A. In: Journal of the American Chemical Society, 137, 2015, 13488--13491 |
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| 2015 | Yao, Guiyang and Pan, Zhengyin and Wu, Chunlei and Wang, Wei and Fang, Lijing and Su, Wu: Efficient synthesis and stereochemical revision of coibamide A. In: Journal of the American Chemical Society, 137, 2015, 13488--13491 |
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| 2015 | Lijing, Fang and Guiyang, Yao and Zhengyin, Pan and Chunlei, Wu and Heng-Shan, Wang and Wu, Su and others: Fully Automated Synthesis of DNA-Binding Py-Im Polyamides Using a Triphosgene Coupling Strategy. 2015, |
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| 2015 | Fang, Lijing and Yao, Guiyang and Pan, Zhengyin and Wu, Chunlei and Wang, Heng-Shan and Burley, Glenn A and Su, Wu: Fully automated synthesis of DNA-binding Py-Im polyamides using a triphosgene coupling strategy. In: Organic Letters, 17, 2015, 158--161 |
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| 2015 | Li, Ya-Jun and Wang, Cai-Yi and Ye, Man-Yi and Yao, Gui-Yang and Wang, Heng-Shan: Novel coumarin-containing aminophosphonatesas antitumor agent: synthesis, cytotoxicity, DNA-binding and apoptosis evaluation. In: Molecules, 20, 2015, 14791--14809 |
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| 2015 | Li, Ya-Jun and Wang, Cai-Yi and Ye, Man-Yi and Yao, Gui-Yang and Wang, Heng-Shan: Novel coumarin-containing aminophosphonatesas antitumor agent: synthesis, cytotoxicity, DNA-binding and apoptosis evaluation. In: Molecules, 20, 2015, 14791--14809 |
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| 2015 | Qu, Hong-En and Huang, Ri-Zhen and Yao, Gui-Yang and Li, Jiu-Ling and Ye, Man-Yi and Wang, Heng-Shan and Liu, Liangxian: Synthesis and pharmacological evaluation of novel bisindole derivatives bearing oximes moiety: Identification of novel proapoptotic agents. In: European Journal of Medicinal Chemistry, 95, 2015, 400--415 |
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| 2015 | Qu, Hong-En and Huang, Ri-Zhen and Yao, Gui-Yang and Li, Jiu-Ling and Ye, Man-Yi and Wang, Heng-Shan and Liu, Liangxian: Synthesis and pharmacological evaluation of novel bisindole derivatives bearing oximes moiety: Identification of novel proapoptotic agents. In: European Journal of Medicinal Chemistry, 95, 2015, 400--415 |
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| 2014 | Liu, Shi-Jun and Liao, Zhi-Xin and Liu, Chao and Yao, Gui-Yang and Wang, Heng-Shan: A new triterpenoid and eremophilanolide from Ligularia przewalskii. In: Phytochemistry Letters, 9, 2014, 11--16 |
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| 2014 | Li, Ya-Jun and Ye, Man-Yi and Huang, Ri-Zhen and Yao, Gui-Yang and Pan, Ying-Ming and Liao, Zhi-Xin and Wang, Heng-Shan: Coumarin-containing aminophosphonates bridged with chiral side chain: Synthesis and influence of chirality on cytotoxicity and DNA binding. In: Medicinal Chemistry Research, 23, 2014, 3144--3156 |
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| 2014 | Yao, Guiyang and Li, Yajun and Zhu, Yongtao and Pan, Yingming and Huang, Fuping and Wang, Hengshan and Liao, Zhixin: Protonation-controlled axial chirality in maleopimaric imides. In: New Journal of Chemistry, 38, 2014, 693--699 |
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| 2014 | Ye, Man-Yi and Yao, Gui-Yang and Pan, Ying-Ming and Liao, Zhi-Xin and Zhang, Ye and Wang, Heng-Shan: Synthesis and antitumor activities of novel $\alpha$-aminophosphonate derivatives containing an alizarin moiety. In: European journal of medicinal chemistry, 83, 2014, 116--128 |
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| 2014 | Ye, Man-Yi and Yao, Gui-Yang and Pan, Ying-Ming and Liao, Zhi-Xin and Zhang, Ye and Wang, Heng-Shan: Synthesis and antitumor activities of novel $\alpha$-aminophosphonate derivatives containing an alizarin moiety. In: European journal of medicinal chemistry, 83, 2014, 116--128 |
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| 2014 | Yao, Gui-yang and Ye, Man-yi and Huang, Ri-zhen and Li, Ya-jun and Pan, Ying-ming and Xu, Qing and Liao, Zhi-Xin and Wang, Heng-shan: Synthesis and antitumor activities of novel rhein $\alpha$-aminophosphonates conjugates. In: Bioorganic \& Medicinal Chemistry Letters, 24, 2014, 501--507 |
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| 2014 | Yao, Gui-yang and Ye, Man-yi and Huang, Ri-zhen and Li, Ya-jun and Pan, Ying-ming and Xu, Qing and Liao, Zhi-Xin and Wang, Heng-shan: Synthesis and antitumor activities of novel rhein $\alpha$-aminophosphonates conjugates. In: Bioorganic \& Medicinal Chemistry Letters, 24, 2014, 501--507 |
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| 2014 | Li, Jian-Fei and Huang, Ri-Zhen and Yao, Gui-Yang and Ye, Man-Yi and Wang, Heng-Shan and Pan, Ying-Ming and Xiao, Jing-Teng: Synthesis and biological evaluation of novel aniline-derived asiatic acid derivatives as potential anticancer agents. In: European Journal of Medicinal Chemistry, 86, 2014, 175--188 |
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| 2014 | Li, Jian-Fei and Huang, Ri-Zhen and Yao, Gui-Yang and Ye, Man-Yi and Wang, Heng-Shan and Pan, Ying-Ming and Xiao, Jing-Teng: Synthesis and biological evaluation of novel aniline-derived asiatic acid derivatives as potential anticancer agents. In: European Journal of Medicinal Chemistry, 86, 2014, 175--188 |
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| 2013 | Huang, Guo-Bao and Wang, Xu and Pan, Ying-Ming and Wang, Heng-Shan and Yao, Gui-Yang and Zhang, Ye: Atom-economical chemoselective synthesis of 1, 4-enynes from terminal alkenes and propargylic alcohols catalyzed by Cu (OTf) 2. In: The Journal of organic chemistry, 78, 2013, 2742--2745 |
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| 2013 | Huang, Guo-Bao and Wang, Xu and Pan, Ying-Ming and Wang, Heng-Shan and Yao, Gui-Yang and Zhang, Ye: Atom-economical chemoselective synthesis of 1, 4-enynes from terminal alkenes and propargylic alcohols catalyzed by Cu (OTf) 2. In: The Journal of organic chemistry, 78, 2013, 2742--2745 |
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| 2013 | Yao, Guiyang and Wei, Jingchen and Dai, Weilong and Yang, Da and Pan, Yingming and Wang, Hengshan: Study on the regioselectivie of Grignard reagent addition reaction of maleopimaric acid trimethyl ester. In: Chinese Journal Of Organic Chemistry, 33, 2013, 138--142 |
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| 2013 | Huang, Xiao-Chao and Wang, Meng and Pan, Ying-Ming and Yao, Gui-Yang and Wang, Heng-Shan and Tian, Xiao-Yan and Qin, Jiang-Ke and Zhang, Ye: Synthesis and antitumor activities of novel thiourea $\alpha$-aminophosphonates from dehydroabietic acid. In: European Journal of Medicinal Chemistry, 69, 2013, 508--520 |
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| 2013 | Huang, Xiao-Chao and Wang, Meng and Pan, Ying-Ming and Yao, Gui-Yang and Wang, Heng-Shan and Tian, Xiao-Yan and Qin, Jiang-Ke and Zhang, Ye: Synthesis and antitumor activities of novel thiourea $\alpha$-aminophosphonates from dehydroabietic acid. In: European Journal of Medicinal Chemistry, 69, 2013, 508--520 |
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| 2013 | Yao, Gui-yang and Ye, Man-yi and Huang, Ri-zhen and Li, Ya-jun and Zhu, Yong-tao and Pan, Ying-ming and Liao, Zhi-Xin and Wang, Heng-shan: Synthesis and antitumor activity evaluation of maleopimaric acid N-aryl imide atropisomers. In: Bioorganic \& Medicinal Chemistry Letters, 23, 2013, 6755--6758 |
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| 2013 | Yao, Gui-yang and Ye, Man-yi and Huang, Ri-zhen and Li, Ya-jun and Zhu, Yong-tao and Pan, Ying-ming and Liao, Zhi-Xin and Wang, Heng-shan: Synthesis and antitumor activity evaluation of maleopimaric acid N-aryl imide atropisomers. In: Bioorganic \& Medicinal Chemistry Letters, 23, 2013, 6755--6758 |
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| 2013 | Ye, Man-Yi and Yao, Gui-Yang and Wei, Jing-Chen and Pan, Ying-Ming and Liao, Zhi-Xin and Wang, Heng-Shan: Synthesis, cytotoxicity, DNA binding and apoptosis of rhein-phosphonate derivatives as antitumor agents. In: International journal of molecular sciences, 14, 2013, 9424--9439 |
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| 2013 | Ye, Man-Yi and Yao, Gui-Yang and Wei, Jing-Chen and Pan, Ying-Ming and Liao, Zhi-Xin and Wang, Heng-Shan: Synthesis, cytotoxicity, DNA binding and apoptosis of rhein-phosphonate derivatives as antitumor agents. In: International journal of molecular sciences, 14, 2013, 9424--9439 |
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