| 2019 | Pierre Fontanillas and Achim Kless and John Bothmer and Joyce Y. Tung and: Genome-wide association study of pain sensitivity assessed by questionnaire and the cold pressor test. 2019, |
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| 2019 | Astrid S. Obrecht and Nicole Urban and Michael Schaefer and Anni Röse and Achim Kless and Jannis E. Meents and Angelika Lampert and Aliaa Abdelrahman and Christa E. Müller and Günther Schmalzing and Ralf Hausmann: Identification of aurintricarboxylic acid as a potent allosteric antagonist of P2X1 and P2X3 receptors. In: Neuropharmacology, 158, 2019, 107749 |
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| 2019 | Achim Kless, Ph.D. Investigating targets for neuropharmacological intervention by molecular dynamics simulations.. In: Biochemical Society transactions, 2019, |
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| 2019 | Matthew McIntyre and Achim Kless and Peter Hein and Mark Field and Joyce Y Tung and: Validity of the Cold Pressor Test and Pain Sensitivity Questionnaire via online self-administration. 2019, |
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| 2018 | Achim Kless, Ph.D. and Juan Zeng and Riccardo Guareschi and Mangesh Damre and Ruyin Cao and Achim Kless and Bernd Neumaier and Andreas Bauer and Alejandro Giorgetti and Paolo Carloni and Giulia Rossetti: Structural Prediction of the Dimeric Form of the Mammalian Translocator Membrane Protein TSPO: A Key Target for Brain Diagnostics. In: International Journal of Molecular Sciences, 2018, |
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| 2017 | Anja Pippel and Michaela Stolz and Ronja Woltersdorf and Achim Kless and Günther Schmalzing and Fritz Markwardt: Localization of the gate and selectivity filter of the full-length P2X7 receptor. In: Proceedings of the National Academy of Sciences, 114, 2017, E2156--E2165 |
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| 2017 | Irena Loryan and Edmund Hoppe and Klaus Hansen and Felix Held and Achim Kless and Klaus Linz and Virginia Marossek and Bert Nolte and Paul Ratcliffe and Derek Saunders and Rolf Terlinden and Anita Wegert and Andr{\'{e}} Welbers and Olaf Will and Margareta Hammarlund-Udenaes: Quantitative Assessment of Drug Delivery to Tissues and Association with Phospholipidosis: A Case Study with Two Structurally Related Diamines in Development. In: Molecular Pharmaceutics, 14, 2017, 4362--4373 |
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| 2017 | Achim Kless, Ph.D. Structural heterogeneity of the \mu-opioid receptor{'}s conformational ensemble in the apo state.. In: Scientific reports, 2017, |
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| 2016 | Achim Kless, Ph.D. Thiol dependent intramolecular locking of Orai1 channels.. In: Scientific reports, 2016, |
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| 2015 | Hausmann, Ralf and Kless, Achim and Schmalzing, Gunther: Key Sites for P2X Receptor Function and Multimerization: Overview of Mutagenesis Studies on a Structural Basis. In: Curr Med Chem, 22, 2015, 799-818 |
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| 2015 | Cong, Xiaojing and Campomanes, Pablo and Kless, Achim and Schapitz, Inga and Wagener, Markus and Koch, Thomas and Carloni, Paolo: Structural determinants for the binding of morphinan agonists to the μ-opioid receptor. In: PLoS One, 10, 2015, e0135998/1-e0135998/15 |
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| 2014 | Schunk, Stefan and Linz, Klaus and Frormann, Sven and Hinze, Claudia and Oberbörsch, Stefan and Sundermann, Bernd and Zemolka, Saskia and Englberger, Werner and Germann, Tieno and Christoph, Thomas and Kögel, Babette- Y. and Schröder, Wolfgang and Harlfinger, Stephanie and Saunders, Derek and Kless, Achim and Schick, Hans and Sonnenschein, Helmut: Discovery of Spiro[cyclohexane-dihydropyrano[3,4-b]indole]-amines as Potent NOP and Opioid Receptor Agonists. In: ACS Medicinal Chemistry Letters, 5, 2014, 851-856 |
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| 2014 | Schunk, Stefan and Linz, Klaus and Hinze, Claudia and Frormann, Sven and Oberbörsch, Stefan and Sundermann, Bernd and Zemolka, Saskia and Englberger, Werner and Germann, Tieno and Christoph, Thomas and Kögel, Babette- Y. and Schröder, Wolfgang and Harlfinger, Stephanie and Saunders, Derek and Kless, Achim and Schick, Hans and Sonnenschein, Helmut: Discovery of a Potent Analgesic NOP and Opioid Receptor Agonist: Cebranopadol. In: ACS Medicinal Chemistry Letters, 5, 2014, 857-862 |
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| 2013 | Saul, Anika and Hausmann, Ralf and Kless, Achim and Nicke, Annette: Heteromeric assembly of P2X subunits. In: Frontiers in Cellular Neuroscience, 7, 2013, 20 |
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| 2013 | Hausmann, Ralf and Guenther, Janka and Kless, Achim and Kuhlmann, Daniel and Kassack, Matthias U. and Bahrenberg, Gregor and Markwardt, Fritz and Schmalzing, Guenther: Salt bridge switching from Arg290/Glu167 to Arg290/ATP promotes the closed-to-open transition of the P2X2 receptor. In: Mol.Pharmacol., 83, 2013, 73-84 |
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| 2012 | Nardi, Antonio and Damann, Nils and Hertrampf, Torsten and Kless, Achim: Advances in targeting voltage-gated sodium channels with small molecules. In: ChemMedChem, 7, 2012, 1712-1740 |
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| 2011 | Wolf, Christian and Rosefort, Christiane and Fallah, Ghada and Kassack, Matthias U. and Hamacher, Alexandra and Bodnar, Mandy and Wang, Haihong and Illes, Peter and Kless, Achim and Bahrenberg, Gregor and Schmalzing, Guenther and Hausmann, Ralf: Molecular determinants of potent P2X2 antagonism identified by functional analysis, mutagenesis, and homology docking. In: Mol.Pharmacol., 79, 2011, 649-661 |
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| 2007 | Eitrich, T. and Kless, A. and Druska, C. and Meyer, W. and Grotendorst, J.: Classification of highly unbalanced CYP450 data of drugs using cost sensitive machine learning techniques. In: J.Chem.Inf.Model., 47, 2007, 92-103 |
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| 2003 | Kless, Achim and Tarkhov, Alexei and Pfoertner, Matthias and Bangov, Ivan: Accelerated processes with data mining development. In: Nachr.Chem., 51, 2003, 1264-1266 |
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| 1999 | Quirmbach, Michael and Kless, Achim and Holz, Jens and Tararov, Vitali and Borner, Armin: Construction of chiral Ti(IV)-Rh(I)-salenophos complexes and their application in the asymmetric hydroformylation of functionalized olefins. In: Tetrahedron: Asymmetry, 10, 1999, 1803-1811 |
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| 1999 | Kless, Achim and Nendel, Maja and Wilsey, Sarah and Houk, K. N.: Origin of the Preference for the Orbital Symmetry Forbidden Stereochemistry of the 1,5-Sigmatropic Shift of Substituted Norcaradienes. In: J.Am.Chem.Soc., 121, 1999, 4524-4525 |
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| 1998 | Houk, K. N. and Wilsey, S. L. and Beno, Brett R. and Kless, Achim and Nendel, Maja and Tian, Jing: Retro-cycloadditions and sigmatropic shifts: The C7H8 and C7H10 potential energy surfaces. In: Pure Appl.Chem., 70, 1998, 1947-1952 |
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| 1998 | Kless, Achim and Holz, Jens and Reinke, Helmut and Borner, Armin: Studies on the formation of uniform eta3-coordinated triphos-Mo(0)-complexes. In: J.Organomet.Chem., 553, 1998, 99-102 |
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| 1997 | Kless, Achim and Boerner, Armin and Heller, Detlef and Selke, Ruediger: Ab Initio Studies of Rhodium(I)-N-Alkenylamide Complexes with cis- and trans-Coordinating Phosphines: Relevance for the Mechanism of Catalytic Asymmetric Hydrogenation of Prochiral Dehydroamino Acids. In: Organometallics, 16, 1997, 2096-2100 |
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| 1996 | Holz, Jens and Kless, Achim and Boerner, Armin: An efficient strategy for the synthesis of new chiral and prochiral trisphosphines. In: Synlett, 1996, 267-269 |
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| 1996 | Kless, Achim and Holz, Jens and Heller, Detlef and Kadyrov, Renat and Selke, Ruediger and Fischer, Christine and Boerner, Armin: Chiral phosphinephosphites having axial and central chirality in asymmetric hydroformylations. In: Tetrahedron: Asymmetry, 7, 1996, 33-36 |
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| 1996 | Kless, A.: Computational Chemistry Using the PC by Donald W. Rogers. In: Z.Phys.Chem.(Munich), 193, 1996, |
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| 1996 | Kless, Achim and Lefeber, Claudia and Spannenberg, Anke and Kempe, Rhett and Baumann, Wolfgang and Holz, Jens and Boerner, Armin: The first chiral early-late heterobimetallic complex - a titanium(IV)-palladium(II) complex based on salenophos. In: Tetrahedron, 52, 1996, 14599-14606 |
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| 1995 | Kless, Achim and Kadyrov, Renat and Boerner, Armin and Holz, Jens and Kagan, Henri B.: A new chiral multidentate ligand for asymmetric catalysis. In: Tetrahedron Lett, 36, 1995, 4601-4602 |
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| 1995 | Boerner, Armin and Kless, Achim and Kempe, Rhett and Heller, Detlef and Holz, Jens and Baumann, Wolfgang: Beta-Alkoxy- and beta-hydroxyalkylphosphines as ligands in the stereoselective hydrogenation - a comparison. In: Chem.Ber., 128, 1995, 767-773 |
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| 1995 | Boerner, Armin and Kless, Achim and Holz, Jens and Baumann, Wolfgang and Tillack, Annegret and Kadyrov, Renat: Complexation of enantiomeric cis- and trans-3-diphenylphosphino-4-hydroxy-tetrahydrofurans with [Rh(COD)2]BF4. In: J.Organomet.Chem., 490, 1995, 213-219 |
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| 1995 | Holz, Jens and Boerner, Armin and Kless, Achim and Borns, Susanne and Trinkhaus, Stephan and Seleke, Ruediger and Heller, Detlef: Hydroxyalkylphosphines in asymmetric hydrogenations. In: Tetrahedron: Asymmetry, 6, 1995, 1973-1988 |
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| 1995 | Boerner, Armin and Holz, Jens and Kless, Achim and Heller, Detlef: Synthesis of hydroxyDIOP ligands and their application in the rhodium-catalyzed asymmetric hydrogenation. In: GIT Fachz.Lab., 39, 1995, 1146-1147 |
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| 1994 | Boerner, Armin and Ward, Jacques and Ruth, Wolfgang and Holz, Jens and Kless, Achim and Heller, Detlef and Kagan, Henri B.: Synthesis and catalytic properties of an acyclic analog of hydroxy norphos. In: Tetrahedron, 50, 1994, 10419-10430 |
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| 1994 | Borner, Armin and Holz, Jens and Kless, Achim and Heller, Detlef and Berens, Ulrich: Synthesis of an optically active hydroxy diphosphine, a new ligand for asymmetric catalysis. In: Tetrahedron Lett, 35, 1994, 6071-6074 |
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